BRS-3 agonist Compound A

CAS No. ——

BRS-3 agonist Compound A( —— )

Catalog No. M17034 CAS No. ——

A potent, selective, orally active bombesin receptor subtype-3 (BRS-3) agonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    BRS-3 agonist Compound A
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent, selective, orally active bombesin receptor subtype-3 (BRS-3) agonist.
  • Description
    A potent, selective, orally active bombesin receptor subtype-3 (BRS-3) agonist with EC50 of 250/100 nM for human/rat BRS-3, resp+H1437+M1438.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Bombesin Receptor
  • Recptor
    Bombesin Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    ——
  • Formula Weight
    428.532
  • Molecular Formula
    C27H28N2O3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    ——
  • Chemical Name
    R-6-benzyl-N-tert-butyl-9-methoxy-7-oxo-6,7-dihydro-5H-dibenzo[c,e]azepine-5-carboxamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Nio Y, et al. Endocrinology. 2017 May 1;158(5):1298-1313.
molnova catalog
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